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Berberine Hydrochloride
API ea Tlhaho

Berberine Hydrochloride

● Berberine hydrochloride ke alkaloid ea tlhaho ea isoquinoline e nkiloeng limela tsa meriana tse kang Coptis chinensis (goldthread) le Phellodendron amurense (sefate sa Amur cork). Jwalo ka motsoako wa bohlokwa o sebetsang meriana ya setso, dipatlisiso tsa sejwalejwale di tiisitse mesebetsi ya yona ya baeloji ya mefuta e mengata, haholoholo ho laoleng metabolism ya glucose le lipid le ho bontsha ditlamorao tsa ho lwantsha dikokwana-hloko. Hangata e bitswa "sebolaya-dikokwana-hloko sa tlhaho sa dimela."

Lebitso la Sehlahisoa: Berberine Hydrochloride

Lebitso la Khemikhale: 5,6-Dihydro-9,10-dimethoxybenzo[g]-1,3-benzodioxolo[5,6-a]quinolizinium chloride

Foromo ea limolek'hule: C₂₀H₁₈ClNO₄

    tlhaloso1

    tlhaloso2

    berberine hcl

    Tlhahisoleseding ea Motheo

    Lebitso la Sehlahisoa: Berberine Hydrochloride

    Lebitso la Khemikhale:5,6-Dihydro-9,10-dimethoxybenzo[g]-1,3-benzodioxolo[5,6-a]quinolizinium chloride

    Foromo ea limolek'hule: C₂₀H₁₈ClNO₄

    Nomoro ea CAS:【 633-65-8】

    Boima ba limolek'hule: 372.822

    Ho qhibiliha ha metsi: E qhibiliha habonolo metsing a belang, e qhibiliha hanyane metsing a batang, 'me e batla e sa qhibilihe ho ethanol e batang, chloroform, le ether.

    Maemo a Boleng: CP2020, JP, E entsoe ke Moreki

    Tlhaloso

    Lintho tsa Teko

    E tloaelehileng

    Berberine Hydrochloride 【633-65-8】

    ≥97.0% ka HPLC

    Tahlehelo ha ho omisoa

    ≤12.0%

    Masalla a ho hotetsa

    ≤0.2%

    Likarolo tsa Bohlokoa

    Melemo ea Mesebetsi e Mengata

    Taolo ea Metabolism: E kenya tshebetsong ditsela tsa AMPK ho tshehetsa taolo ya tswekere le mafura mading, e loketse batho ba nang le lefu la tswekere kapa botenya.

    Sebolaya-mafu le se Loantšang ho ruruha: E thibela likokoana-hloko tse kang E. coli le Staphylococcus aureus, e thusa ho tšoaetso ea mala.

    Bophelo bo Botle ba Mala: E fetola microbiota ea mala, e fokotsa letšollo le ho se sile hantle ha lijo.

    Tšimoloho ea Tlhaho

    E tsoa litlameng tsa meriana, e kopanyang katleho ea setso le netefatso ea saense.

    Bohloeki bo Phahameng

    Tlhoekiso e tsoetseng pele e netefatsa bohloeki ba ≥98% bakeng sa katleho le botsitso bo botle.

    antibacterial ea road-spectrum

    Khahlanong le mefuta e fapaneng ea libaktheria tse ntle tsa Gram le Gram (mohlala, Shigella, Escherichia coli, Staphylococcus aureus, Hemolytic streptococcus, pneumococcus, typhoid bacilli, jj.)

    Litlamorao tsa meriana Boholo bo botala

    Berberine hydrochloride e na le phello e pharaletseng ea antibacterial, 'me mokhoa oa eona oa ketso o kenyelletsa haholo-holo:

    1. Ho sitisa metabolism ea baktheria: Ho thibela ts'ebetso ea oxidation le decarboxylation ea pyruvate, e leng khokahano ea lipakeng tsa metabolism ea tsoekere ea baktheria.

    2. Thibela ho ikatisa ha DNA ea baktheria. E ama metabolism ea nucleic acid ea baktheria 'me e sitisa tlhahiso ea lintho tsa bona tsa lefutso.

    3. Tšenyo sebopehong sa baktheria: E na le phello e senyang lera la sele la baktheria mme e ama mosebetsi oa tsona oa thibelo.

    4. Taolo ea ho thibela ho ruruha le ea sesole sa 'mele: E na le phello e itseng ea ho thibela ho ruruha 'me e ka fokotsa likarabo tsa ho ruruha mala; Lithuto tse ling li boetse li bontša hore e na le phello ea taolo mosebetsing oa sesole sa 'mele mala.

    5. E hlabang le e thibelang letšollo: E na le phello e hlabang lera la mala 'me e fokotsa ho ntšoa ha mokelikeli oa mala.

    Phellodendron amurense

    Tekanyo le Tsamaiso

    1. Batho ba baholo: 100–300 mg, makhetlo a 2-3 ka letsatsi kamora lijo (buisana le ngaka bakeng sa tekanyo e nepahetseng).

    2. Lithibelo: Ha ea lokela basali ba bakhachane kapa bakuli ba nang le hemolytic jaundice; qoba ho e sebelisa ka nako e le 'ngoe le meriana e fokotsang tsoekere kapa lithibela-mafu (ho hlokahala tlhokomelo ea bongaka).

    Profaele ea Polokeho​

    Lithuto tsa bongaka li bontša litla-morao tse fokolang (mohlala, ho ruruha kapa ho pipitleloa ka linako tse ling) ka tekanyo e khothaletsoang, ntle le chefo ea hepatorenal. Tšebeliso ea nako e telele e lokela ho kenyelletsa tlhokomelo ea bophelo bo botle nako le nako.

    Ka kopo nthomelle imeile 'me u ka fumana tse ling tseo u li batlang.

    Joalo ka sehlahisoa sa Theko, Tlhaloso, MOA, MSDS, Chate ea Phallo, Lintlha tsa ho Paka, Nako ea ho Romela, Nako ea Tefo, Tšebeletso ea Kamora Thekiso jj.

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